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RGH 896 - Radiprodil

 

 

CAS 496054-87-6

C21H20FN3O4  MW 397.41 

Purity: 99%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1434   

 

Qty1: 5 mg (research sample) / €115  $150

Qty2: 10 mg (research sample) / €165  $215

Qty3: 50 mg (research sample) / €660  $858

 

Qty4: on request contract research synthesis

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:

 

Orally active and selective NMDA NR2B antagonist; a potential therapeutic agent in treatment of neuropathic pain and possibly other chronic pain conditions. It blocks pain signaling without interacting with other NMDA receptor subtypes thus potentially improving therapeutic index and side effect profile.

 

References: online

 

 

 

 

Chemical Name: 1-Piperidineacetamide, N-(2,3-dihydro-2-oxo-6-benzoxazolyl)-4-[(4-fluorophenyl)methyl]-α-oxo

 

RGH 896 - Radiprodil | NMDA NR2B antagonist | Axon Medchem | Axon 1434 | RGH896

 

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

axonmedchem.com © 2009

 

Axon Ligands In This Field:

 

CP 101606 | NMDA antagonist

Ifenprodil | NMDA antagonist

Eliprodil | NMDA antagonist

N20C | NMDA antagonist

Gavestinel | Glycine antagonist

Radiprodil | NMDA antagonist

Ro 25-6981 | NMDA antagonist

 

CNQX | AMPA/kanaite antagonist

DNQX | AMPA/kainate antagonist

GYKI 53655 | AMPA antagonist

YM-90K | AMPA antagonist

 

MPEP | mGluR5 antagonist

Fenobam | mGluR5 antagonist

YM 298198 | mGlu1 antagonist

LY 367385 | mGlu1a antagonist