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Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

 

 

 

  

DH 97

 

CAS 343263-95-6

C22H26N2O  MW 334.47

Purity: 98%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1351

 

Qty1: 10 mg / €95  $124

 

Qty2: 50 mg / €335  $436

 

Qty3: on request

 

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Biological Activity:

 

Melatonin antagonist; MT2 selective

 

References: online 1, 2

 

MT Teh & D Sugden. Comparison of the structure-activity relationships of melatonin receptor agonists and antagonists: lengthening the N-acyl side-chain has differing effects on potency on Xenopus melanophores. Naunyn Schmiedebergs Arch. Pharmacol. 1998, 358, 522.
 

KN Ting et al. Molecular and pharmacological evidence for MT1 melatonin receptor subtype in the tail artery of juvenile Wistar rats. Br. J. Pharmacol. 1999, 127, 987.

 

 

Chemical Name: Pentanoic acid [2-(2-benzyl-1H-indol-3-yl)-ethyl]-amide; or N-Pentanoyl-2-benzyltryptamine

 

DH 97 | Melatonin MT2 antagonist | Axon Medchem | Axon 1351 - DH97 - DH-97

axonmedchem.com © 2011

 

Axon Ligands In The Field:

 

AH 001 | Melatonin agonist

AH 002 | Melatonin agonist

DH 97 | Melatonin MT2 antagonist

Luzindole | Melatonin antagonist 

 

 

 

 

 

 

 

 

Axon Ligands TM

 

Research chemicals for biological study. Some high-profile ligands could be provided under terms of contract research synthesis.