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Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

 

 

 

  

GR 103691

 

 

 

 

CAS 162408-66-4

C30H35N3O3  MW 485.63

Purity: 99%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1347

 

Qty1: 10 mg / €95  $124

 

Qty2: 50 mg / €335  $436

 

Qty3: on request

 

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Biological Activity:

 

Dopamine D3 receptor antagonist.

 

References:

 

Audinot et al. A comparative in vitro and in vivo pharmacological characterization of the novel dopamine D3 receptor antagonists (+)-S 14297, nafadotride, GR 103,691 and U 99194. J. Pharmacol. Exp. Ther. 1998, 287, 187.

 

 

Chemical Name: 4'-Acetyl-biphenyl-4-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide

 

GR 103691 | D3 antagonist | Axon Medchem | Axon 1347 | GR103691

axonmedchem.com © 2011

 

Axon DRD3 related ligands: e.g.

 

7-hydroxy-DPAT | D3 agonist

(R)-(+)-7-OH-DPAT | D3 agonist

(±)-PD 128907 | D3 agonist

(+)-PD 128907 | D3 agonist

ST 198 | D3 antagonist

U 99194 | D3 antagonist

GR 103691 | D3 antagonist

 

 

 

Axon Ligands TM

 

Research chemicals for biological studies. Some high-profile samples could be provided under terms of contract research synthesis.