Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

B-HT 958 dihydrochloride

CAS 83718-64-3

C14H14ClN3S.2HCl

MW 366.74

Purity: 99 %

Ordering Information:

Cat. No. Axon 1337

Qty1: 10 mg / €95  $124

Qty2: 50 mg / €295  $384

Qty3: on request

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Biological Activity:   Dopamine D2 receptor agonist, α2-adrenoceptor partial agonist   References: online ref 1, 2, 3, 4   MJ Brown and D Harland. B-HT 958 lowers blood pressure and heart rate in the rat through stimulation of dopamine receptors. Br. J. Pharmacol. 1986, 87(2), 361–370.   G Cichini et al. B-HT 920 and B-HT 958: Presynaptic effects on electrically evoked 3H-dopamine release from slices of rat nucleus accumbens. Naunyn-Schmiedeberg's Arch. Pharmacol. 1987, 335, 28-31.   L Pichler et al. B-HT 958, a new α-adrenoceptor agonist with a high pre/postsynaptic activity ratio. Naunyn-Schmiedeberg's Arch. Pharmacol. 1982, 320, 2, 110-114.   Chemical Name: 6-(4-chlorobenzyl)-2-amino-5,6,7,8-tetrahydro-4H-thiazolo-[4,5-d]azepine

B-HT 958 | alpha-2 partial and D2 agonist | Axon Medchem | Axon 1337 | B-HT958 - BHT 958

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Axon Ligands in the area:

Atipamezole | α2 antagonist

B-HT 920 | α2 and D2 agonist

B-HT 933 | α2 agonist

B-HT 958 | α2 partial & D2 agonist

Efaroxan | α2 antagonist

ST-91 | α2 agonist