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Iodophenpropit dihydrobromide

 

 

CAS 143407-29-8

C15H19IN4S.2HBr  

MW 576.13

Purity: 98%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1328

 

Qty1: 10 mg / €119  $155

 

Qty2: 50 mg / €479  $623

 

Qty3: on request

 

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Biological Activity:

 

Potent and selective histamine H3 receptor antagonist

 

References: online 1, 2

 

Leurs et al. Evaluation of the receptor selectivity of the H3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5-HT3 receptor revealed. Br. J. Pharmacol. 1995, 116(4): 2315–2321.

 

Jansen et al. Characterisation of the binding of the first selective radiolabelled histamine H3 receptor antagonist, [125I]-iodophenpropit, to rat brain. r. J. Pharmacol. 1994, 113, 355.

 

 

Chemical Name: N-[2-(4-Iodophenyl)ethyl]-S-[3-(4(5)-imidazolyl)propyl] isothiourea dihydrobromide

 

Iodophenpropit (IPP) | H3 antagonist | Axon Ligands | Axon Medchem | Axon 1328

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Histamine Receptor (HR) Ligands available: e.g.

 

ABT 239 | H3 antagonist

Amthamine | H2 agonist

Clobenpropit | H3 antagonist

Dimaprit | H2 agonist

Fexofenadine | H1 antagonist

Imetit | H3 agonist

Immepip | H3 agonist

Immethridine | H3 agonist

Iodophenpropit | H3 antagonist

JNJ 7777120 | H4 antagonist

JNJ 10191584 | H4 antagonist

Loratadine | H1 antagonist

4-Methylhistamine | H4 agonist

PF 3654746 | H3 antagonist