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Biological Activity:
Potent and selective histamine H3 receptor antagonist
References: online 1, 2
Leurs et al. Evaluation of the receptor selectivity of the H3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5-HT3 receptor revealed. Br. J. Pharmacol. 1995, 116(4): 2315–2321.
Jansen et al. Characterisation of the binding of the first selective radiolabelled histamine H3 receptor antagonist, [125I]-iodophenpropit, to rat brain. r. J. Pharmacol. 1994, 113, 355.
Chemical Name: N-[2-(4-Iodophenyl)ethyl]-S-[3-(4(5)-imidazolyl)propyl] isothiourea dihydrobromide
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