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Immepip dihydrobromide

 

 

CAS 164391-47-3

C9H15N3.2HBr 

MW 327.06

Purity: 98%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1326

 

Qty1: 10 mg / €105  $137

 

Qty2: 50 mg / €425  $553

 

Qty3: on request

 

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Biological Activity:

 

Potent histamine H3 receptor agonist; also with affinity at H4 receptor.

 

References:

 

Y Lamberty et al. H3 agonist immepip markedly reduces cortical histamine release, but only weakly promotes sleep in the rat. Pharmacol. Res. 2003,48, 192-198.

 

Liuet al. Cloning and pharmacological characterization of a fourth histamine receptor (H4) expressed in bone marrow. Mol. Pharmacol. 2001, 59 420.

 

 

Chemical Name:4-(1H-Imidazol-4-ylmethyl)piperidine dihydrobromide

 

Immepip | H3 agonist | Axon Medchem | Axon 1326

 

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Histamine Receptor (HR) Ligands available: e.g.

 

ABT 239 | H3 antagonist

Amthamine | H2 agonist

Clobenpropit | H3 antagonist

Dimaprit | H2 agonist

Fexofenadine | H1 antagonist

Imetit | H3 agonist

Immepip | H3 agonist

Immethridine | H3 agonist

Iodophenpropit | H3 antagonist

JNJ 7777120 | H4 antagonist

JNJ 10191584 | H4 antagonist

Loratadine | H1 antagonist

4-Methylhistamine | H4 agonist

PF 3654746 | H3 antagonist