Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

CGS 21680 hydrochloride

CAS 124182-57-6 (HCl)

120225-54-9 (parent)

C23H29N7O6.HCl  MW 499.53

Purity: >98 %

Ordering Information:

Cat. No. Axon 1319      Prime Source

Qty1: 5 mg / €98  $128

Promotion: 2 x 5 mg @ €150  $195

Qty2: 25 mg / €340  $442

Promotion: 2 x 25 mg @ €550  $715

Qty3: on request (* in stock of grams)

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

Contact us for payment and tech support.

Biological Activity:   Selective A2A adenosine receptor agonist   References: online 1, 2, 3   CA Mayer et al. Adenosine A2A receptors mediate GABAergic inhibition of respiration in immature rats. J. Appl. Physiol. 2006,100(1), 91-97.   N Levens et al. Renal actions of a new adenosine agonist CGS 21680A selective for the A2 receptor. J. Pharmacol. Exp. Ther. 1991, 257, 1005-1012.   JW Phillis. The selective adenosine A2 receptor agonist, CGS 21680, is a potent depressant of cerebral cortical neuronal activity. Brain Res. 1990, 509, 328-330.     Chemical Name: 3-(4-{2-[6-Amino-9-((2R,3R,4S,5S)-5-ethylcarbamoyl-3,4-dihydroxy-tetrahydro-furan-2-yl)-9H-purin-2-ylamino]-ethyl}-phenyl)-propionic acid

CGS 21680 | A2A agonist | Axon Medchem | Axon 1319 | CGS21680 - CGS 21680A

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

axonmedchem.com © 2012

Axon Adenosine Receptor (AR) Ligands: e.g.

CGS 21680 | A2A agonist

KW 6002 | A2A antagonist

SCH 442416 | A2A antagonist

SCH 58261 | A2A antagonist

ADAC | A1 agonist

2-Chloroadenosine | A1/2A ago.

GR 79236 | A1 agonist

SDZ WAG 994 | A1 agonist

Rolofylline | A1 antagonist