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Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

 

 

 

  

SKF 83566 hydrobromide

 

 

CAS 99295-33-7 (parent)

108179-91-5 (HBr salt)

C17H18BrNO.HBr MW 413.15 

Purity: 99%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1236

 

Qty1: 10 mg / €70  $91

 

Qty2: 50 mg / €280  $364

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:

 

Selective dopamine D1-like receptor antagonist

 

References:

 

R Pedrosa et al. Defective D1-like receptor-mediated inhibition of the Cl/HCO3 exchanger in immortalized SHR proximal tubular epithelial cells. Am. J. Physiol. Renal. Physiol. 2004, 286, F1120-F1126.

 

Meyeret al. Effects of dopamine D1 antagonists SCH23390 and SK&F83566 on locomotor activities in rats. Pharmacol. Biochem. Behav. 1993, 44, 429.

 

 

 

Chemical Name:8-Bromo-2,3,4,5-tetrahydro-3-methyl-5-phenyl-1H-3-benzazepin-7-ol hydrobromide

 

SKF-83566 | D1 antagonist | Axon Medchem | Axon 1236 | SKF83566

axonmedchem.com © 2012

 

Axon Ligands in the area:

 

NNC 756 | D1 antagonist

SKF-83566 | D1 antagonist

Molindone | D2 antagonist

ST 148 | D2 antagonist 

ST 198 | D3 antagonist

U 99194 | D3 antagonist

GR 103691 | D3 antagonist

Amisulpride | D2/D3 antagonist

Aripiprazole | D2 partial agonist

Sertindole | D2/5-HT2 antagonist

Olanzapine | D1/2/4 antagonist