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Naloxone Benzoylhydrazone

CAS 119630-94-3

C26H27N3O4  MW 445.51

Purity: >98%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1230   Prime Source

 

Qty1: 10 mg / €85  $111

 

Qty2: 50 mg / €335  $436

 

Qty3: on request

 

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or by fax to: +31-50-3600390.

 

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Biological Activity:

 

Agonist for κ3 opioid receptors; antagonist for ORL1 and μ opioid receptors.

 

References: online 1, 2

 

MA Gistrak et al. Pharmacological actions of a novel mixed opiate agonist

/antagonist: Naloxone benzoylhydrazone. J. Pharmacol. Exp. Ther. 1989, 251, 469-476.

 

D Paul et al. Naloxone benzoylhydrazone (NalBzoH) analgesia. J. Pharmacol. Exp. Ther. 1990, 255, 769-774.

 

 

Chemical Name: [(5α)-4,5-Epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]hydrazide benzoic acid

 

Naloxone Benzoylhydrazone | opioid ligand | Axon Medchem | Axon 1230

 

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Opioid Receptor Ligands:

 

nor-BNI | k opioid antagonist

β-FNA | μ opioid antagonist

GNTI | k opioid antagonist

Nalmefene | opioid antagonist

Naloxonazine | opioid antagonist

Naloxone Benzoylhydrazone

 

ADL 5859 | δ opioid agonist

Fedotozine | k opioid agonist

SNC 80 | δ opioid agonist

U 50488 | k opioid agonist

 

BAN ORL 24 | NOP antagonist

JTC 801 | NOP antagonist

SB 612111 | NOP antagonist