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Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

 

 

 

  

GNTI  -  6'-Guanidinonaltrindole dihydrochloride

 

 

 

C27H29N5O3.2HCl

MW 544.48

Purity: >98%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1226

 

Qty1: 5 mg / €95  $124

 

Qty2: 25 mg / inquire

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

Contact us for payment and tech support.

 

Biological Activity:

 

kappa opioid antagonist

 

References:

 

CT Qi et al. Effect of GNTI, a kappa opiid receptoe antagonist, on MK-801-induced hyperlocomotion and stereotypy in mice. Acta Pharmacol. Sin. 2006, 27(11), 1401-8.

 

 

 

 

Chemical Name:6''-Guanidinyl-17-(cyclopropylmethyl)-6,7-dehydro-4,5a- epoxy-3,14-dihydroxy-6,7-2',3'-indolomorphinan dihydrochloride

 

GNTI | kappa opioid antagonist | Axon Medchem | Axon 1226

axonmedchem.com © 2012

 

Axon Opioid Receptor Ligands:

 

nor-BNI | k opioid antagonist

β-FNA | μ opioid antagonist

GNTI | k opioid antagonist

Nalmefene | opioid antagonist

Naloxonazine | opioid antagonist

Naloxone Benzoylhydrazone

 

ADL 5859 | δ opioid agonist

Fedotozine | kopioid agonist

SNC 80 | δ opioid agonist

U 50488 | k opioid agonist

 

BAN ORL 24 | NOP antagonist

JTC 801 | NOP antagonist

SB 612111 | NOP antagonist