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Biological Activity:
kappa opioid antagonist
References:
CT Qi et al. Effect of GNTI, a kappa opiid receptoe antagonist, on MK-801-induced hyperlocomotion and stereotypy in mice. Acta Pharmacol. Sin. 2006, 27(11), 1401-8.
Chemical Name:6''-Guanidinyl-17-(cyclopropylmethyl)-6,7-dehydro-4,5a- epoxy-3,14-dihydroxy-6,7-2',3'-indolomorphinan dihydrochloride
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