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AM 281

CAS 202463-68-1

C21H19Cl2IN4O2 MW 557.22

Purity: 99 %

Ordering Information:

Cat. No. Axon 1219

Qty1: 10 mg / €95  $124

Qty2: 50 mg / €305  $397

Qty3: on request

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Biological Activity:   Potent and selective CB1 cannabinoid receptor antagonist/inverse agonist   References:   F Molina-Holgado et al. Neuroprotective effects of the synthetic cannabinoid HU-210 in primary cortical neurons are mediated by phosphatidylinositol 3-kinase/AKT signaling. Mol. Cell. Neurosci. 2005, 28, 189-194.   AN Gifford et al. Effect of the cannabinoid receptor SPECT agent, AM 281, on hippocampal acetylcholine release from rat brain slices. Neurosci. Lett. 1997,  238, 84-86.   Chemical Name: 1-(2,4-Dichloro-phenyl)-5-(4-iodo-phenyl)-4-methyl-1H-pyrazole-3-carboxylic acid morpholin-4-ylamide

AM 281 | CB1 antagonist | Axon Medchem | Axon 1219 | AM281

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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