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β-Funaltrexamine hydrochloride

β-FNA hydrochloride

CAS 72786-10-8

C25H30N2O6.HCl  MW 490.98

Purity: 98%

 

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1213

 

Qty1: 10 mg / inquire

 

Qty2: 50 mg / inquire

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:

 

Selective irreversible μ opioid receptor antagonist

 

References: online 1

 

JH Broadbear et al. Methocinnamox is a potent long-lasting and selective antagonist of morphine-mediated antinociception in the mouse: comparison with clocinnamox, beta-funaltrexamine and beta-chlornaltrexamine. J. Pharmacol. Exp. Ther. 2000, 294, 933.

 

 

Chemical Name: (E)-4-[[(5α,6β)-17-(Cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxymorphinan-6-yl]amino]-4-oxo-2-butenoic acid methyl ester hydrochloride

 

beta-Funaltrexamine | μ opioid antagonist | Axon Medchem | Axon 1213 | beta-FNA

axonmedchem.com © 2011

 

Axon Opioid Receptor Ligands:

 

nor-BNI | k opioid antagonist

β-FNA | μ opioid antagonist

GNTI | k opioid antagonist

Nalmefene | opioid antagonist

Naloxonazine | opioid antagonist

Naloxone Benzoylhydrazone

 

ADL 5859 | δ opioid agonist

Fedotozine | kopioid agonist

SNC 80 | δ opioid agonist

U 50488 | k opioid agonist

 

BAN ORL 24 | NOP antagonist

JTC 801 | NOP antagonist

SB 612111 | NOP antagonist