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Clobenpropit dihydrobromide

 

 

 

CAS 145231-45-4 (free base)

145231-35-2 (2HBr)

C14H17ClN4S.2HBr  MW 470.65 

Purity: 99%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1209

 

Qty1: 10 mg / 90  $117

Promotion: 2 x 10 mg @ 135  $176

Qty2: 50 mg / 270  $351

Promotion: 2 x 50 mg @ 405  $527

Qty3: on request

 

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or by fax to: +31-50-3600390.

 

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Biological Activity:

 

Potent histamine H3 receptor antagonist

 

References:

 

Yokoyamaet al. Clobenpropit (VUF-9153), a new histamine H3 receptor antagonist, inhibits electrically induced convulsions in mice. Eur. J. Pharmacol. 1994, 260, 23.

 

 

Chemical Name: 1-(4-Chloro-benzyl)-2-[3-(1H-imidazol-4-yl)-propyl]-isothiourea dihydrobromide

 

Clobenpropit | H3 antagonist | Axon Medchem | VUF 9153 | Axon 1209

 

Axon Ligands TM

Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Histamine Receptor (HR) Ligands available: e.g.

 

ABT 239 | H3 antagonist

Amthamine | H2 agonist

Clobenpropit | H3 antagonist

Dimaprit | H2 agonist

Fexofenadine | H1 antagonist

Imetit | H3 agonist

Immepip | H3 agonist

Immethridine | H3 agonist

Iodophenpropit | H3 antagonist

JNJ 7777120 | H4 antagonist

JNJ 10191584 | H4 antagonist

Loratadine | H1 antagonist

4-Methylhistamine | H4 agonist

PF 3654746 | H3 antagonist