PK 11195 | Benzodiazepine Antagonist | Axon Ligands | Axon Medchem

Chemistry Service Platform - CRO in Medicinal Chemistry

PK 11195

CAS 85532-75-8

C21H21ClN2O MW 352.86

Purity: >98%

Ordering Information:

Cat. No. Axon 1208

Qty1: 10 mg / €65 $85

Qty2: 50 mg / €195 $254

Qty3: on request

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

Biological Activity:

Peripheral benzodiazepine antagonist.

References:

Klegeris, A., et al., Inhibitory action of 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide (PK 11195) on some mononuclear phagocyte functions. Biochem. Pharmacol. 2000, 59, 1305-1314.

Wala, E.P., et al., Pharmacokinetics of the peripheral benzodiazepine receptor antagonist, PK 11195, in rats. The effect of dose and gender. Pharmacol. Res. 2000, 41, 461-468.

Chemical Name: 1-(2-Chloro-phenyl)-isoquinoline-3-carboxylic acid sec-butyl-methyl-amide

PK 11195 | Benzodiazepine Antagonist | Axon Medchem | Axon 1208 | PK11195

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Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.