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GBR 12783 dihydrochloride

 

 

CAS 67469-75-4 (HCl)

67469-57-2 (free base)

C28H32N2O.2HCl  MW 485.47

Purity: 99%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1203

 

Qty1: 10 mg / €85  $111

 

Qty2: 50 mg / €285  $371

 

Qty3: on request

 

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Biological Activity:

 

Potent and selective inhibitor of dopamine uptake

 

References:

 

Bonnet and Constentin. GBR 12783, a potent and selective inhibitor of dopamine uptake: biochemical studies in vivo and ex vivo. Eur. J. Pharmacol. 1986, 121 199.

 

Do-Rego et al. Evidence for the sequential formation of two complexes between an uptake inhibitor, GBR 12783 [1-[2-(diphenylmethoxy)ethyl]-4-(3-phenyl-2-propenyl)piperazine], and the neuronal transporter of dopamine. J. Neurochem. 1999, 72, 396.

 

 

Chemical Name: 1-(2-Benzhydryloxy-ethyl)-4-((E)-3-phenyl-allyl)-piperazine dihydrochloride

 

GBR 12783 | Dopamine uptake inhibitor | Axon Medchem | Axon 1203 | GBR12783

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Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.