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nor-Binaltorphimine dihydrochloride

CAS 113158-35-3

105618-26-6 (parent)

C40H43N3O6.2HCl  MW 734.72

Purity: >98%

 

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1163

 

Qty1: 10 mg / inquire

 

Qty2: 50 mg / inquire

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:

 

Potent and selective kappa opioid receptor antagonist

 

References:

 

SD Mague et al. Antidepressant-like effects of kappa-opioid receptor antagonists in the forced swim test in rats. J. Pharmacol Exp. Ther. 2003, 305(1), 323-30.
 

MJ Picker et al. Opioids and rate of positively reinforced behavior: III. Antagonism by the long-lasting kappa antagonist norbinaltorphimine. Behav Pharmacol 1996, 7(6), 495-504.

 

 

Chemical Name:

 

nor-Binaltorphimine | k opioid antagonist | Axon Medchem | Axon 1163 | nor-BNI

 

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

axonmedchem.com © 2011

 

Axon Opioid Receptor Ligands:

 

ADL 5859 | δ opioid agonist

Fedotozine | kopioid agonist

SNC 80 | δ opioid agonist

U 50488 | k opioid agonist

 

nor-BNI | k opioid antagonist

β-FNA | μ opioid antagonist

GNTI | k opioid antagonist

Nalmefene | opioid antagonist

Naloxonazine | opioid antagonist

Naloxone Benzoylhydrazone

 

BAN ORL 24 | NOP antagonist

JTC 801 | NOP antagonist

SB 612111 | NOP antagonist