GMC 1-165 | Clozapine analogue | Axon Ligands | Axon Medchem

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GMC 1-165

C18H20N4O MW 308.39

Purity: >98%

Ordering Information:

Cat. No. Axon 1152

Qty1: 10 mg / 135 $176

Qty2: 50 mg / inquire

Qty3: on request

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

Biological Activity:

Analogue of clozapine (Axon 1146); devoid of DA affinities but with affinities at 5-HT2A/2C and hM1 receptors.

References:

Liao, Y. et al. Synthesis and pharmacological evaluation of triflate-substituted analogues of Clozapine: Identification of a novel atypical neuroleptic. J. Med. Chem. 1997, 40, 4146-4153.

Liao, Y. et al. New sulfonyloxy piperazinyl-dibenzo-azapines as potential atypical antipsychotics: chemistry and pharmacological evaluation. J. Med. Chem. 1999, 42, 2235-2244.

Chemical Name: 11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepin-2-ol

GMC 1-165 | Clozapine analogue | Axon Medchem | Axon 1152 | GMC1-165 - GMC 1165