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Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

 

 

 

  

GMC 2-83

 

CAS 183140-98-9

C19H18F3N3O4S  MW 441.43

Purity: >98%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1150

 

Qty1: 10 mg / €145  $189

 

Qty2: 50 mg / inquire

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

Contact us for our product range and services.

 

Biological Activity:

 

Atypical antipsychotic lack of muscarinic activity

 

References: onlineref 1, 2

 

Y Liao et al. New sulfonyloxy piperazinyl-dibenzo-azapines as potential atypical antipsychotics: chemistry and pharmacological evaluation. J. Med. Chem. 1999, 42, 2235-2244.

 

Y Liao et al. Synthesis and pharmacological evaluation of triflate-substituted analogues of Clozapine: Identification of a novel atypical neuroleptic. J. Med. Chem. 1997, 40, 4146-4153.

 

D Jackson, H Wikström, Y Liao. Is clozapine an (partial) agonist at both dopamine D1 and D2 receptors? Psychopharmacology 1998, 138, 213-214.

 

 

Chemical Name: Trifluoro-methanesulfonic acid 11-(4-methyl-piperazin-1-yl)-dibenzo[b,f][1,4]oxazepin-2-yl ester

 

GMC 2-83 | Atypical Antipsychotic | Axon Medchem | Axon 1150 | GMC2-83 | GMC 283

 

Axon Ligands TM

Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

axonmedchem.com © 2011

 

Axon Atypical Antipsychotics available: e.g.

 

Amisulpride (Axon 1381)

Aripiprazole (Axon 1143)

Asenapine (Axon 1503)

Bifeprunox (Axon 1508)

Clozapine (Axon 1146)

GMC 1-169 (Axon 1148)

GMC 2-83 (Axon 1150)

GMC 61-39 (Axon 1149)

Iloperidone (Axon 1493)

Olanzapine (Axon 1298)

Quetiapine (Axon 1354)

Risperidone (Axon 1454)

Sertindole (Axon 1141)

Thio-aripiprazole (Axon 1144)

Ziprasidone (Axon 1446)

 

Typical Antipsychotic:

Isoclozapine (Axon 1147)

 

Clozapine Analogues:

GMC 1-116 (Axon 1151)

GMC 1-165(Axon 1152)