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GMC 61-39

 

CAS 234113-94-1

C19H18ClF3N4O3S  MW 474.89

Purity: >98%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1149

 

Qty1: 10 mg / inquire

 

Qty2: 50 mg / inquire

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

Contact us for our product range and services.

 

Biological Activity:

 

Clozapine-like atypical antipsychotic

 

References: online ref 1, 2

 

Liao, Y. et al. Synthesis and pharmacological evaluation of triflate-substituted analogues of Clozapine: Identification of a novel atypical neuroleptic. J. Med. Chem. 1997, 40, 4146-4153.

 

Liao, Y. et al. New sulfonyloxy piperazinyl-dibenzo-azapines as potential atypical antipsychotics: chemistry and pharmacological evaluation. J. Med. Chem. 1999, 42, 2235-2244.

 

Jackson, D; Wikström, H; Liao, Y. Is clozapine an (partial) agonist at both dopamine D1 and D2 receptors? Psychopharm. 1998, 138, 213-214.

 

 

 

 

Chemical Name: Trifluoro-methanesulfonic acid 8-chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepin-2-yl ester

 

GMC 61-39 | Atypical Antipsychotic | Axon Medchem | Axon 1149 | GMC61-39 | GMC 6139

axonmedchem.com © 2011

 

Axon Atypical Antipsychotics available: e.g.

 

Amisulpride (Axon 1381)

Aripiprazole (Axon 1143)

Asenapine (Axon 1503)

Bifeprunox (Axon 1508)

Clozapine (Axon 1146)

GMC 1-169 (Axon 1148)

GMC 2-83 (Axon 1150)

GMC 61-39 (Axon 1149)

Iloperidone (Axon 1493)

Olanzapine (Axon 1298)

Quetiapine (Axon 1354)

Risperidone (Axon 1454)

Sertindole (Axon 1141)

Thio-aripiprazole (Axon 1144)

Ziprasidone (Axon 1446)

 

"Typical Antipsychotic":

Isoclozapine (Axon 1147)

 

Clozapine Analogues:

GMC 1-116 (Axon 1151)

GMC 1-165 (Axon 1152)