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Eltoprazine hydrochloride

DU 28853

 

CAS 98206-09-8 (HCl)

98224-03-4 (free base)

C12H16N2O2.HCl 

MW 256.73

Purity: 99%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1142

 

Qty1: 10 mg / €82  $107

 

Qty2: 50 mg / €322  $419

 

Qty3: on request

 

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Biological Activity:

 

5-HT1A/1Bagonist and 5-HT2C receptor antagonist

 

References: online 1

 

Eltoprazine. WHO Drug Information 1(2): 98, 1987.

 

G Griebel et al. Serenics fluprazine (DU 27716) and eltoprazine (DU 28853) enhance neophobic and emotional behaviour in mice. Psychopharmacology 1990, 102, 498-502.

 

DR. Cherek et al. Acute effects of eltoprazine on aggression and point-mantained responding of normal male participants: Phase I study. Exp. Clin. Psychopharmacol. 1995, 3/3, 287-293.

 

 

Chemical Name: 1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazine hydrochloride

 

Eltoprazine | 5-HT1A/1B agonist, 5-HT2C antagonist  | Axon Medchem | Axon 1142 | DU28853

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Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.