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BX 912

 

 

CAS702674-56-4

C20H23BrN8O 

MW 471.36

Purity: >98%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1130     Prime Source

 

Qty1: 2 mg (research sample) / €90  $117

Qty2: 5 mg (research sample) / €135  $176

Qty3: 25 mg (research sample) / €485  $631

 

Qty4: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:

 

Inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1).

 

References: online ref 1

 

RI Feldman et al. Novel Small Molecule Inhibitors of 3-Phosphoinositide-dependent Kinase-1. J. Biol. Chem., 2005, 280, 20, 19867-19874.
 

C Peifer and DR Alessi. Small-Molecule Inhibitors of PDK1. ChemMedChem. 2008, 3 (10),  Review. [online]

 

 

 

Chemical Name: Pyrrolidine-1-carboxylic acid (3-{5-bromo-4-[2-(1H-imidazol-4-yl)-ethylamino]-pyrimidin-2-ylamino}-phenyl)-amide

 

BX 912 | PDK1 inhibitor | Axon Medchem | Axon 1130 | BX912

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Ligands In The Field:

 

BX 912 | PDK1 inhibitor

BX 795 | TBK1/PDK1 inhibitor

PS 48 | PDK1 activator

 

 

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