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Biological Activity:
Inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1).
References: online ref 1
RI Feldman et al. Novel Small Molecule Inhibitors of 3-Phosphoinositide-dependent Kinase-1. J. Biol. Chem., 2005, 280, 20, 19867-19874.
C Peifer and DR Alessi. Small-Molecule Inhibitors of PDK1. ChemMedChem. 2008, 3 (10), Review. [online]
Chemical Name: Pyrrolidine-1-carboxylic acid (3-{5-bromo-4-[2-(1H-imidazol-4-yl)-ethylamino]-pyrimidin-2-ylamino}-phenyl)-amide
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