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Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

 

 

 

  

Molindone hydrochloride   

EN-1733 A  

CAS 15622-65-8 (HCl)

7416-34-4 (free base)

C16H24N2O2·HCl  MW 312.83

Purity: 99 %

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1101

 

Qty1: 10 mg / €85  $111

 

Qty2: 50 mg / €205  $267

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:

 

D2 dopamine receptor antagonist; MAO inhibitor; a therapeutic antipsychotic, used in the treatment of schizophrenia; Reduction of body weight reported. Terminal plasma half-life after oral administration about 6½ hours.

 

 

References: online

 

A Bagnall et al. Molindone for schizophrenia and severe mental illness. Cochrane Database Syst. Rev. 2007, 1, CD002083. [online]

 

DB Allison et al. Antipsychotic-induced weight gain: a comprehensive research synthesis. Am. J. Psychiatry 1999, 156(11), 1686–1696. [abstract] [online]

 

 

 

Chemical Name: 3-Ethyl-2-methyl-5-morpholin-4-ylmethyl-1,5,6,7-tetrahydro-indol-4-one hydrochloride

 

Molindone | D2 antagonist - MAO inhibitor | Axon Medchem | Axon 1101

axonmedchem.com © 2011

 

Axon Dopamine Ligands: e.g.

5-hydroxy-DPAT | D2 agonist

(S) 5-hydroxy-DPAT | D2 agonist

R(-)-NPA | D2 agonist

RU 24213 | D2 agonist

(+)-PHNO | D2 agonist

PPHT - N-0434 | D2 agonist

Molindone | D2 antagonist

ST 148 | D2 antagonist

 

ABT 724 | D4 agonist

CP 226269 | D4 agonist

 

7-hydroxy-DPAT | D3 agonist

(R)-(+)-7-OH-DPAT | D3 agonist

(±)-PD 128907 | D3 agonist

(+)-PD 128907 | D3 agonist

ST 198 | D3 antagonist

U 99194 | D3 antagonist

GR 103691 | D3 antagonist

 

S-(+)-Dinapsoline | D1 agonist

NNC 776 | D1 antagonist

SKF-83566 | D1 antagonist

N-0426 | DA agonist

N 0734 | DA agonist  

Rotigotine - N-0437 | DA agonist

(-)-Rotigotine | DA agonist

Piribedil | Dopamine agonist

TL 99 | Dopamine agonist

TL 102 | Dopamine agonist

TL 232 | Dopamine agonist