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SB 258741 hydrochloride

CAS 201038-58-6 (free base)

C18H29N3O2S  MW 351.51

Purity: >98%

Ordering Information:

Cat. No. Axon 1100

Qty1: 5 mg (research sample) / €115  $150

Qty2: 25 mg (research sample) / €415  $540

Qty3: on request

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Biological Activity:   Serotonin 5-HT7 antagonist.   References: online ref 1, 2   Porset B.SB-258741: a 5-HT7 receptor antagonist of potential clinical interest. CNS Drug Rev. 2002, 8(1), 90-100.   Mahe B et al. Differential inverse agonist efficacies of SB-258719, SB-258741 and SB-269970 at human recombinant serotonin 5-HT7 receptors. Eur J Pharmacol. 2004, 495(2-3), 97-102.     Chemical Name:4-Methyl-1-{2-[(R)-1-(toluene-3-sulfonyl)-pyrrolidin-2-yl]-ethyl}-piperidine hydrochloride

SB-258741 | 5-HT7 antagonist | Axon Medchem | SB258741 | Axon 1100

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