SB 216641 | 5-HT1B antagonist | Axon Ligands | Axon Medchem

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SB 216641 hydrochloride

CAS 193611-67-5 (HCl)

170230-39-4 (parent)

C₂₈H₃₀N₄O₄.HCl MW 523.03

Purity: >98 %

Soluble in water and DMSO

Ordering Information:

Cat. No. Axon 1085

Qty1: 10 mg / 135 $176

Promotion: 2 x 10 mg @ 180 $234

Qty2: 50 mg / 540 $702

Promotion: 2 x 50 mg @ 780 $1014

Qty3: on request

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

Biological Activity:

Selective human 5-HT1B antagonist

References:

Schlicker et al. Effects of selective h5-HT_1B (SB-216641) and 5-HT_1D (BRL-15572) receptor ligands on guinea pig and human 5-HT auto- and heteroreceptors. Naunyn-Schmied. Arch. Pharmacol. 1997, 356, 321.

Chemical Name: N-[3-[3-(Dimethylamino)ethoxy]-4-methoxyphenyl]-2'-meth yl-4'-(5-methyl-1,2,4-oxadiazol-3-yl)-[1,1'-biphenyl]-4 -carboxamide hydrochloride

SB 216641 | 5-HT1B antagonist | Axon Medchem | SB216641 | Axon 1085