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Biological Activity:
Very potent and selective 5-HT1B/1D antagonist
References: online 1
Liao et al. New selective and potent 5-HT1B/1D or 5-HT1B antagonists: chemistry and pharmacological evaluation of GR127935-like compounds. J. Med. Chem. 2000, 43, 517-525.
Clitherow et al. Evolution of a novel series of [(N,N-dimethylamino)propyl]- and piperazinylbenzalides as the first selective 5-HT1D antagonists. J. Med. Chem. 1994, 37, 2253.
Chemical Name: 2-Methyl-biphenyl-4,4'-dicarboxylic acid 4-amide 4'-{[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide}
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