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(±)-PD 128907 hydrochloride

PD-125530

 

 

CAS 123594-64-9

C14H19NO3·HCl  MW 285.77

Purity: >98%

(trans-racemic)

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1072

 

Qty1: 5 mg / 115  $150

 

Qty2: 25 mg / 415  $540

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:

 

Selective D3 dopamine receptor agonist.

 

Its more active enantiomer is trans-(+)-PD-128907 (Axon 1073) and less active enantiomer is (-)-PD 128907 (Axon 1074).

 

References: online ref 1, 2

 

Pugsley et al. Neurochemical and functional characterization of the preferentially selective dopamine D3 agonist PD 128907. J. Pharmacol. Exp. Ther. 1995, 275 1355.

 

Chemical Name: trans-(+/-)-3,4a,4,10b-Tetrahydro-4-propyl-2H,5H-[1]benzopyrano-[4,3-b]-1,4-oxazin-9-ol hydrochloride; also as PD-125,530

 

(±)-PD 128907 | Selective D3 agonist | Axon Medchem | Axon 1072 | (±)-PD128907, (±)-PD 128,907

axonmedchem.com © 2011

 

DRD3 related ligands: e.g.

 

7-hydroxy-DPAT | D3 agonist

(R)-(+)-7-OH-DPAT | D3 agonist

(±)-PD 128907 | D3 agonist

(+)-PD 128907 | D3 agonist

ST 198 | D3 antagonist

U 99194 | D3 antagonist

GR 103691 | D3 antagonist

 

 

 

Axon Ligands TM

 

Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.