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U 99194 maleate

CAS 234757-41-6

 82668-33-5 (free base)

C₁₇H₂₇NO₂.C₄H₄O₄  MW 393.48

Purity: >98 %

Ordering Information:

Cat. No. Axon 1069

Qty1: 10 mg / €80  $104

Qty2: 50 mg / €320  $416

Qty3: on request

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Biological Activity:   Selective and potent D3 antagonist with a 30-fold preference for the dopamine D3 vs D2 receptor.   References:   Kling-Petersen, et al., Effects on locomotor activity after local application of D3 preferring compounds in discrete areas of the rat brain. J. Neural Transm. 1995, 102, 209-220.   Audinot et al. A comparative in vitro and in vivo pharmacological characterization of the novel dopamine D3 receptor antagonists (+)-S 14297, nafadotride, GR 103,691 and U 99194. J. Pharmacol. Exp. Ther. 1998, 287 187.       Chemical Name: (5,6-Dimethoxy-indan-2-yl)-dipropyl-amine maleate; or 5,6-Dimethoxy-2-(di-n-propylamino)indan maleate; [153570-58-2]

U-99194 | D3 antagonist | Axon Medchem | U99194 | Axon 1069

axonmedchem.com © 2011

Axon DRD3 related ligands: e.g.

7-hydroxy-DPAT | D3 agonist

(R)-(+)-7-OH-DPAT | D3 agonist

(±)-PD 128907 | D3 agonist

(+)-PD 128907 | D3 agonist

ST 198 | D3 antagonist

U 99194 | D3 antagonist

GR 103691 | D3 antagonist

NNC 756 | D1 antagonist

SKF-83566 | D1 antagonist

Molindone | D2 antagonist

ST 148 | D2 antagonist

Olanzapine | D1/2/4 antagonist... 

Axon Ligands ^TM

Research chemicals for biological studies. Some high-profile samples could be provided under terms of contract research synthesis.