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PPHT hydrochloride - N-0434

 

 

CAS 71787-90-1 (HCl)

87857-27-0 (free base)

C21H27NO.HCl  MW 345.91

Purity: >98%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1035

 

Qty1: 10 mg / €125  $163

 

Qty2: 50 mg / €450  $585

 

Qty3: on request

 

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or by fax to: +31-50-3600390.

 

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Biological Activity:

 

Very Potent and specific D2 agonist

 

References: online ref 1, 2, 3

 

Van der Weide, J. et al., , Pharmacological profiles of three new, potent and selective dopamine receptor agonists: N-0434, N-0437 and N-0734. Eur. J. Pharmacol.125, 273-282, (1986).

 

Seeman, P., et al., Dopamine D2 receptor binding sites for agonists. A tetrahedral model. Mol. Pharmacol.28, 391, (1985).

 

 

 

 

 

 

 

 

Chemical Name: (±)-2-(N-Phenethyl-N-propyl)amino-5-hydroxytetralin hydrochloride

 

PPHT | D2 agonist | Axon Medchem | Axon 1035 | N-0434
Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Dopamine Ligands: e.g.

 

S-(+)-Dinapsoline | D1 Agonist

GR 103691 | D3 antagonist

5-hydroxy-DPAT | D2 agonist

(S) 5-hydroxy-DPAT | D2 agonist

7-hydroxy-DPAT | D3 agonist

(R)-(+)-7-OH-DPAT | D3 agonist

Molindone | D2 antagonist

N-0426 | DA agonist

N 0734 | DA agonist  

NNC 776 | D1 antagonist

R(-)-NPA | D2 agonist

Rotigotine - N-0437 | DA agonist

(-)-Rotigotine | DA agonist

RU 24213 | D2 agonist

(±)-PD 128907 | D3 agonist

(+)-PD 128907 | D3 agonist

(+)-PHNO | D2 agonist

Piribedil | Dopamine agonist

PPHT - N-0434 | D2 agonist

SKF-83566 | D1 antagonist

ST 148 | D2 antagonist

ST 198 | D3 antagonist

TL 99 | Dopamine agonist

TL 102 | Dopamine agonist

TL 232 | Dopamine agonist

U 99194 | D3 antagonist